Evaluation of Oxetan-3-ol, Thietan-3-ol, and Derivatives Thereof as Bioisosteres of the Carboxylic Acid Functional Group | ACS Medicinal Chemistry Letters
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Interleukin-17A Peptide Aptamers with an Unexpected Binding Moiety Selected by cDNA Display under Heterogenous Conditions | ACS Medicinal Chemistry Letters
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Expanding the Medicinal Chemist Toolbox: Comparing Seven C(sp2)–C(sp3) Cross-Coupling Methods by Library Synthesis | ACS Medicinal Chemistry Letters
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Introducing the Tellurophene-Appended BODIPY: PDT Agent with Mass Cytometry Tracking Capabilities | ACS Medicinal Chemistry Letters
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Structural Rigidification of N-Aryl-pyrroles into Indoles Active against Intracellular and Drug-Resistant Mycobacteria | ACS Medicinal Chemistry Letters
Systematic Investigation of the Permeability of Androgen Receptor PROTACs | ACS Medicinal Chemistry Letters
Development of Potent and Selective Janus Kinase 2/3 Directing PG–PROTACs | ACS Medicinal Chemistry Letters
Design, Synthesis, and Evaluation of Donepezil-Like Compounds as AChE and BACE-1 Inhibitors | ACS Medicinal Chemistry Letters
Profiling and Application of Photoredox C(sp3)–C(sp2) Cross-Coupling in Medicinal Chemistry | ACS Medicinal Chemistry Letters
Cannabinoids from Cannabis sativa L.: A New Tool Based on HPLC–DAD–MS/MS for a Rational Use in Medicinal Chemistry | ACS Medicinal Chemistry Letters
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